Makarov LaboratoryMakarovLab

intellectual property

Patents

The laboratory patent archive follows research from chemical concept and synthesis to protected molecular classes and preparation methods.

patent archive

Patents

NumberRU 2815974

Year2024

Method for preparing (+)-(12R,13AR,13BS*)-2,3,5,6,12,13,13A,13B-octahydro-1H-indolo[3,2,1-de]pyrido[3,2,1-ij]naphthyridin-12-ol

Makarov V. A, Riabova O. B, Lepeshkin A. Yu.

Open

NumberWO 2023128786

Year2023

New antiviral triazole derivatives, their synthesis and their use for treatment of mammalian viral infections

Makarov V. A, Riabova O. B, Lane T. R, Ekins S.

Open

NumberRU 2756587

Year2021

2-acetamido-6-hydroxybenzothiophene derivatives and pharmaceutically acceptable salts thereof with antiviral activity

Makarov V. A, Zarubaev V. V.

Open

NumberRU 2675240

Year2018

Pyranoindoles with antitubercular activity

Makarov V. A, Lepeshkin A. Yu, Monakhova N. S, Salina E. G.

Open

NumberWO 2017069661

Year2017

Pyrimidyl-di(diazaspiro-alkanes) with antiviral activity

Makarov V. A, Nesterenko V. G, Bolgarin R. N, Novoselova E. A.

Open

NumberWO 2016151011

Year2016

2-Homopiperazine-1-yl-4H-1,3-benzothiazine-4-one derivatives and process for the preparation of 2-(homo)piperazine 1,3-benzothiazine-4-one hydrochlorides(in English)

Stewart C, Makarov V. A.

Open

NumberWO 2015167368

Year2015

4,6-Di(3,12-diaza-6,9-diazoniadispiro[5.2.5.2]hexadecan-1-yl)-2-methyl-5-nitropyrimidine tetrachloride dihydrochloride hexahydrate for the treatment of herpetic infection and a topical pharmaceutical composition

Makarov V. A, Monakhova N. S, Riabova O. B.

Open

NumberRU 2566818

Year2015

Method for preparing (±)N-[1-(4-fluorophenyl)-2-(1-ethylpiperidin-4-yl)ethyl]-4-nitrobenzamide or pharmaceutically acceptable salts thereof

Makarov V. A.

Open

NumberRU 2487132

Year2013

Derivatives of cyclic 5-nitropyridin-2-yl-thioalkenyl-4-dithiocarbamates with antifungal activity and their use

Makarov V. A, Surovtsev V. V.

Open

NumberWO 2013053942

Year2013

4-amino-3-phenylamino-6-phenylpyrazolo[3,4-d]pyrimidine derivatives, their manufacture and their use as antiviral active substances

Макаров В. А, Wutzler P, Schmidtke M.

Open

NumberWO 2012066518

Year2012

2-Piperazin-1-yl-4H-1,3-benzothiazin-4-one derivatives and their use for the treatment of mammalian infections

Makarov V, Stewart C.

Open

NumberWO 2011132070

Year2011

Process for the preparation of 2-amino-substituted 1,3-benzothiazine-4-ones

Makarov V. A.

Open